Discovery of Bis-Imidazoline Derivatives as New CXCR4 Ligands

The chemokine receptor CXCR4 and its ligand CXCL12 regulate leukocyte trafficking, homeostasis and functions and are potential therapeutic targets in many diseases such as HIV-1 infection and cancers.Here, we identified new CXCR4 ligands in the CERMN chemical library using a FRET-based high-throughput screening assay.These are bis-imidazoline compo

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